Concepedia

Design of (N)-methanocarba adenosine 5′-uronamides as species-independent A3 receptor-selective agonists

Artem Melman, Zhan‐Guo Gao, Deepmala Kumar, Tina C. Wan, Elizabeth Gizewski, John A. Auchampach, Kenneth A. Jacobson

Bioorganic & Medicinal Chemistry Letters · 2008 · 45 citations · 29 references

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29

2-Substitution of N6-Benzyladenosine-5'-uronamides Enhances Selectivity for A3 Adenosine Receptors

Hea O. Kim, Xiao-duo Ji, Suhaib M. Siddiqi et al. · Journal of Medicinal Chemistry · 1994 · 204 citations · Full text

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A physiological role of the adenosine A <sub>3</sub> receptor: Sustained cardioprotection

Bruce T. Liang, Kenneth A. Jacobson · Proceedings of the National Academy of Sciences · 1998 · 201 citations · Full text

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The A3 Adenosine Receptor Is Highly Expressed in Tumor <b> <i>versus</i> </b> Normal Cells

Lea Madi, Avivit Ochaion, Lea Rath‐Wolfson et al. · Clinical Cancer Research · 2004 · 191 citations · Full text

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A<sub>3</sub>Adenosine Receptor Activation Triggers Phosphorylation of Protein Kinase B and Protects Rat Basophilic Leukemia 2H3 Mast Cells from Apoptosis

Zhenhai Gao, Bingsheng Li, Yuan‐Ji Day et al. · Molecular Pharmacology · 2001 · 132 citations

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Methanocarba Analogues of Purine Nucleosides as Potent and Selective Adenosine Receptor Agonists

Kenneth A. Jacobson, Xiao‐duo Ji, An‐Hu Li et al. · Journal of Medicinal Chemistry · 2000 · 122 citations · Full text

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