Concepedia

Synthesis and biological activity of selective pipecolic acid-based TNF-α converting enzyme (TACE) inhibitors

Michael A. Letavic, Matt Z. Axt, John T. Barberia, Thomas J. Carty, Dennis E. Danley, Kieran F. Geoghegan, Nadia S. Halim, Lise R. Hoth, Ajith V. Kamath, Ellen R. Laird,

Bioorganic & Medicinal Chemistry Letters · 2002 · 75 citations · 8 references

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8

A metalloproteinase disintegrin that releases tumour-necrosis factor-α from cells

Roy A. Black, Charles T. Rauch, Carl J. Kozlosky et al. · Nature · 1997 · 3.1K citations

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Cloning of a disintegrin metalloproteinase that processes precursor tumour-necrosis factor-α

Marcia L. Moss, S.-L. Catherine Jin, Marcos E. Milla et al. · Nature · 1997 · 1.6K citations

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Crystal structure of the catalytic domain of human tumor necrosis factor-α-converting enzyme

K. Maskos, C. Fernandez-Catalan, Robert Huber et al. · Proceedings of the National Academy of Sciences · 1998 · 384 citations · Full text

Crystal structures of MMP-1 and -13 reveal the structural basis for selectivity of collagenase inhibitors.

Michelle F. Browner, Brett Lovejoy, Anthony Welch et al. · Nature Structural Biology · 1999 · 248 citations

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A High Throughput Fluorogenic Substrate for Interstitial Collagenase (MMP-1) and Gelatinase (MMP-9)

D. Mark Bickett, M.D. Green, Judd Berman et al. · Analytical Biochemistry · 1993 · 107 citations

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