Selective mono- and di-N-alkylation of aromatic amines with alcohols and acylation of aromatic amines using Ph3P/DDQ

The Use of Diethyl Azodicarboxylate and Triphenylphosphine in Synthesis and Transformation of Natural Products

Oyo Mitsunobu · Synthesis · 1981 · 4.1K citations

Natural Sciences, Biochemistry, Chemistry +8

Amide bond formation and peptide coupling

Christian Montalbetti, Virginie M. Falque · Tetrahedron · 2005 · 1.7K citations

Natural Sciences, Chemistry, Organic Chemistry +11

Reductive Amination of Aldehydes and Ketones with Sodium Triacetoxyborohydride. Studies on Direct and Indirect Reductive Amination Procedures¹

Ahmed F. Abdel‐Magid, Kenneth G. Carson, Bruce D. Harris et al. · The Journal of Organic Chemistry · 1996 · 1.5K citations

Natural Sciences, Chemistry, Catalysis +10

1-Hydroxy-7-azabenzotriazole. An efficient peptide coupling additive

Louis A. Carpino · Journal of the American Chemical Society · 1993 · 1.5K citations

Natural Sciences, Chemistry, Pharmacology +7

Copper-Catalyzed Coupling of Alkylamines and Aryl Iodides:  An Efficient System Even in an Air Atmosphere

Fuk Yee Kwong, Artis Klapars, Stephen L. Buchwald · Organic Letters · 2002 · 504 citations

Natural Sciences, Chemistry, Catalysis +11