MCPP but not TFMPP is an antagonist at cardiac 5HT3 receptors

Identification of serotonin M-receptor subtypes and their specific blockade by a new class of drugs

B. P. Richardson, G. Engel, P. Donatsch et al. · Nature · 1985 · 842 citations

Psychiatry, Medicine, Psychotropic Medication +9

The pharmacology and function of 5-HT3receptors

B. P. Richardson, G. Engel · Trends in Neurosciences · 1986 · 385 citations

Molecular Pharmacology, Signal Transduction, Molecular Physiology +7

Relative efficacies of piperazines at the phosphoinositide hydrolysis-linked serotonergic (5-HT-2 and 5-HT-1c) receptors.

P. Jeffrey Conn, Elaine Sanders‐Bush · Journal of Pharmacology and Experimental Therapeutics · 1987 · 220 citations

[3H]Quipazine labels 5-HT3 recognition sites in rat cortical membranes

Stephen J. Peroutka, Anne Hamik · European Journal of Pharmacology · 1988 · 128 citations

Neurophysiology, Rat Cortical Membranes, Medicine +7

5-HT1 and 5-HT2: binding characteristics of some quipazine analogs

Richard A. Glennon, R. M. Slusher, Robert A. Lyon et al. · Journal of Medicinal Chemistry · 1986 · 87 citations · Full text