A short and convenient chemoenzymatic synthesis of both enantiomers of 3-phenylGABA and 3-(4-chlorophenyl)GABA (Baclofen)

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Quantitative analyses of biochemical kinetic resolutions of enantiomers

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Basic Neurochemistry: Molecular, Cellular, and Medical Aspects

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Enantioselective Michael Addition of Nitromethane to α,β-Enones Catalyzed by Chiral Quaternary Ammonium Salts. A Simple Synthesis of (<i>R</i>)-Baclofen

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The biological activity of d-baclofen (Lipresal®)

H.‐R. Olpe, Henri Demieville, V. Baltzer et al. · European Journal of Pharmacology · 1978 · 211 citations

Biological Activity, Medicinal Chemistry, Biochemistry +3