Bioorganic & Medicinal Chemistry · 2006 · 46 citations · 45 references
MedicineMedicinal ChemistryPharmacologyDrug DesignMolecular PharmacologyPharmacodynamicsAnalgesic PharmacologyDrug-receptor InteractionsOpioid AnalgesicsOpioid PharmacologyReceptor PharmacologySteric EffectsFentanyl AnaloguesOpioid PharmacodynamicsOpioid Receptor AgonistsOpioid Receptor BindingOpioid Receptor ModulatorsSteric BulkSteric-electronic Interactions
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Requirement of Rigid-Body Motion of Transmembrane Helices for Light Activation of Rhodopsin
David Farrens, Christian Altenbach, Ke Yang et al. · Science · 1996 · 1.2K citations
Pharmacological characterization of the cloned kappa-, delta-, and mu-opioid receptors.
K Raynor, Hyesik Kong, Yong Chen et al. · Molecular Pharmacology · 1994 · 663 citations · Full text