Concepedia

Structure–activity relationship (SAR) investigations of substituted imidazole analogs as TRPV1 antagonists

Vijay Gore, Vu V., Rami Tamir, Narender R. Gavva, James Treanor, Mark H. Norman

Bioorganic & Medicinal Chemistry Letters · 2007 · 28 citations · 12 references

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12

Impaired Nociception and Pain Sensation in Mice Lacking the Capsaicin Receptor

Michael J. Caterina, Andreas Leffler, Annika B. Malmberg et al. · Science · 2000 · 3.5K citations

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Vanilloid receptor-1 is essential for inflammatory thermal hyperalgesia

John B. Davis, Julie Gray, Martin J. Gunthorpe et al. · Nature · 2000 · 1.8K citations

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Direct activation of capsaicin receptors by products of lipoxygenases: Endogenous capsaicin-like substances

Sun Wook Hwang, Hawon Cho, Jiyeon Kwak et al. · Proceedings of the National Academy of Sciences · 2000 · 1K citations

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The endogenous lipid anandamide is a full agonist at the human vanilloid receptor (hVR1)

D Smart, Martin J. Gunthorpe, Jeffrey C. Jerman et al. · British Journal of Pharmacology · 2000 · 772 citations · Full text

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Simple, Efficient Catalyst System for the Palladium-Catalyzed Amination of Aryl Chlorides, Bromides, and Triflates

John P. Wolfe, Hiroshi Tomori, Joseph P. Sadighi et al. · The Journal of Organic Chemistry · 2000 · 683 citations

, , +16