Concepedia

Exploration of the structure–activity relationship of the diaryl anilide class of ligands for translocator protein—potential novel positron emitting tomography imaging agents

Harry Wadsworth, Paul A. Jones, Wai-Fung Chau, Clare Durrant, Véronique Morisson-Iveson, Joanna Passmore, Dennis M. O’Shea, Duncan Wynn, Imtiaz Ahmed Khan, Andrew Black,

Bioorganic & Medicinal Chemistry Letters · 2012 · 11 citations · 10 references

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10

Mixed-Affinity Binding in Humans with 18-kDa Translocator Protein Ligands

David R. Owen, Roger N. Gunn, Eugenii A. Rabiner et al. · Journal of Nuclear Medicine · 2010 · 354 citations · Full text

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DPA-714, a New Translocator Protein–Specific Ligand: Synthesis, Radiofluorination, and Pharmacologic Characterization

Michelle L. James, Roger Fulton, Johnny Vercoullie et al. · Journal of Nuclear Medicine · 2008 · 273 citations · Full text

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Kinetic analysis in healthy humans of a novel positron emission tomography radioligand to image the peripheral benzodiazepine receptor, a potential biomarker for inflammation

Masahiro Fujita, Masao Imaizumi, Sami S. Zoghbi et al. · NeuroImage · 2007 · 213 citations · Full text

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Method for measuring the logarithm of the octanol–water partition coefficient by using short octadecyl–poly(vinyl alcohol) high-performance liquid chromatography columns

Stephen F. Donovan, Mark C Pescatore · Journal of Chromatography A · 2002 · 192 citations

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PET imaging with [11C]PBR28 can localize and quantify upregulated peripheral benzodiazepine receptors associated with cerebral ischemia in rat

Masao Imaizumi, Hyun Ju Kim, Sami S. Zoghbi et al. · Neuroscience Letters · 2006 · 174 citations

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