RSC Advances · 2013 · 11 citations · 24 references
PharmacyChemistryMedicinal ChemistryDrug DiscoveryOrganic ChemistrySynthetic Medicinal ChemistryDiversity-oriented SynthesisHeterocycle SynthesisHeterocyclic ChemistryHeterocyclic CompoundsMacrocycle SynthesisOrganic SynthesisAsymmetric Heterocycle SynthesisBicyclononyne ChemistryHeterocycle FunctionalizationHeterocyclic Medicinal ChemistryIndole ChemistryIndole SynthesisMedicinal Chemistry ApplicationsMedicinal Heterocycles
A facile process for the synthesis of highly substituted bicyclo[4.1.0]heptenones via Corey–Chaykovsky reaction of quinone monoketals is presented. The obtained products were employed to functionalize 3-position of indoles providing compounds which might have potential use in medicinal chemistry.
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