European Journal of Organic Chemistry · 2013 · 28 citations · 33 references
Natural SciencesChemistryMedicinal ChemistryCatalysisOrganic ChemistryHeterocycle SynthesisHeterocyclic ChemistryOrganic SynthesisC - H Bond FunctionalizationHeterocycle FunctionalizationPyrazole ChemistryPyrazole SynthesisRoom-temperature Synthesis
Abstract A mild and efficient method for the direct alkenylation of 5‐pyrazoles by Pd‐catalyzed C–H bond activation is described. The reaction smoothly proceeds at room temperature to provide products in up to 92 % yield.
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