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On the Use of Five-Membered Heterocycles in Peptide Chemistry*
15
Citations
0
References
1985
Year
Medicinal ChemistryActivated AmidesBiochemistryMedicineDrug DiscoveryNatural SciencesPeptide LibraryN-acyl DerivativesPeptide SynthesisOrganic ChemistryPeptide SciencePeptide ChemistryPharmacologyDerivative (Chemistry)Synthetic ChemistryBiomolecular Engineering
N-Acyl derivatives of 2-benzoxaolethiol, 2-benzothiazolethiol and 2-benzimidazolethiol are proposed for use both as efficient acylating agents for the synthesis of N-benzyloxycarbonyl and N-fluorenylmethyloxycarbonyl amino acid derivatives and as activated amides for the synthesis of peptides.