Concepedia

Structure-activity relationship of N-methyl-N-aralkyl-peptidylamines as novel N-type calcium channel blockers

Lain‐Yen Hu, R. Todd Ryder, Michael Rafferty, David Dooley, Joann J. Geer, Susan M. Lotarski, George P. Miljanich, Elizabeth Millerman, David M. Rock, Sally J. Stoehr,

Bioorganic & Medicinal Chemistry Letters · 1999 · 22 citations · 6 references

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6

Selective N-type neuronal voltage-sensitive calcium channel blocker, SNX-111, produces spinal antinociception in rat models of acute, persistent and neuropathic pain.

S. Scott Bowersox, T Gadbois, Tejinder Singh et al. · Journal of Pharmacology and Experimental Therapeutics · 1996 · 276 citations

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Mitochondrial dysfunction after experimental and human brain injury and its possible reversal with a selective N-type calcium channel antagonist (SNX-lll)

Bon H. Verweij, Paul Muizelaar, Federico C. Viñas et al. · Neurological Research · 1997 · 150 citations

, , +17

Anticonvulsant effects of some calcium entry blockers in DBA/2 mice

Giovambattista De Sarro, Brian S. Meldrum, Giuseppe Nisticò · British Journal of Pharmacology · 1988 · 142 citations · Full text

, , +14

Selective N-Type Calcium Channel Antagonist Omega Conotoxin MVIIA Is Neuroprotective Against Hypoxic Neurodegeneration in Organotypic Hippocampal-Slice Cultures

Ashley K. Pringle, Christopher D. Benham, Lulu Sim et al. · Stroke · 1996 · 95 citations

, , +17

Selective blockade of N-type voltage-sensitive calcium channels protects against brain injury after transient focal cerebral ischemia in rats

S. Scott Bowersox, Tejinder Singh, Robert R. Luther · Brain Research · 1997 · 47 citations

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