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Efficient InCl<sub>3</sub>/H<sub>2</sub>O-Catalyzed One-Pot Stereoselective Synthesis of<i>cis</i>-2-Methyl-4-amido-1,2,3,4-tetrahydroquinoline Derivatives
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2011
Year
Diversity Oriented SynthesisDerivatives2,4-Disubstituted TetrahydrouinolinesCis DiastereoselectivityAromatic AminesOrganic ChemistryStereoselective SynthesisChemistryHeterocycle ChemistryPharmacologyDerivative (Chemistry)Synthetic Chemistry
Abstract Various cis-2-methyl-4-amido-1,2,3,4-tetrahydroquinoline derivatives were synthesized efficiently by reacting aromatic amines and N-vinyl caprolactam or N-vinyl pyrrolidone in the presence of indium trichloride in an aqueous medium in good to excellent yields. These 2,4-disubstituted tetrahydrouinolines showed cis diastereoselectivity.
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