Concepedia

Differentiation of in vitro transcriptional repression and activation profiles of selective glucocorticoid modulators

Steven W. Elmore, John K. Pratt, Michael J. Coghlan, Yue Mao, Brian E. Green, David D. Anderson, Michael A. Stashko, Chun Wel Lin, Douglas L. Falls, Masaki Nakane,

Bioorganic & Medicinal Chemistry Letters · 2004 · 57 citations · 22 references

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22

Antitumor promotion and antiinflammation: Down-modulation of AP-1 (Fos/Jun) activity by glucocorticoid hormone

Carsten Jonat, Hans J. Rahmsdorf, Kun-Koo Park et al. · Cell · 1990 · 1.6K citations

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Transcriptional interference between c-Jun and the glucocorticoid receptor: Mutual inhibition of DNA binding due to direct protein-protein interaction

Hsin‐Fang Yang‐Yen, Jean‐Claude Chambard, Yu-Lin Sun et al. · Cell · 1990 · 1.6K citations

, , +14

Crystal Structure of the Glucocorticoid Receptor Ligand Binding Domain Reveals a Novel Mode of Receptor Dimerization and Coactivator Recognition

Randy K. Bledsoe, Valerie G. Montana, Thomas B. Stanley et al. · Cell · 2002 · 815 citations · Full text

, , +17

Glucocorticoids and insulin resistance: old hormones, new targets

Robert Andrews, Brian R. Walker · Clinical Science · 1999 · 266 citations

, , +16

A Novel Antiinflammatory Maintains Glucocorticoid Efficacy with Reduced Side Effects

Michael J. Coghlan, Peer B. Jacobson, Ben Lane et al. · Molecular Endocrinology · 2003 · 221 citations

, , +17