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Synthesis, SAR and evaluation of [1,4′]-bipiperidinyl-4-yl-imidazolidin-2-one derivatives as novel CCR5 antagonists

David M. Rotstein, Stephen D. Gabriel, Nicole Manser, L. K. FILONOVA, Fernando Padilla, Surya Sankuratri, Changhua Ji, André deRosier, Marianna Dioszegi, Gabrielle Heilek,

Bioorganic & Medicinal Chemistry Letters · 2010 · 12 citations · 3 references

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Orally Bioavailable Competitive CCR5 Antagonists

Gebhard Thoma, François Nuninger, Marc Schaefer et al. · Journal of Medicinal Chemistry · 2004 · 30 citations · Full text

Assessing hERG Channel Inhibition Using PatchXpress

Justin Q. Ly, Gordon Shyy, Dinah Misner · Clinics in Laboratory Medicine · 2007 · 25 citations

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Anti-HIV-1 entry optimization of novel imidazopiperidine-tropane CCR5 antagonists

Justin T. Ernst, Russell Dahl, Christopher Lum et al. · Bioorganic & Medicinal Chemistry Letters · 2007 · 18 citations · Full text

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