Publication | Open Access

Evaluation of secondary amide replacements in a series of CCR5 antagonists as a means to increase intrinsic membrane permeability. Part 1: Optimization of gem-disubstituted azacycles

Medicinal ChemistryMedicineMembrane TransportPeptoidSecondary Amide ReplacementsCcr5 AntagonistsIntrinsic Membrane PermeabilityPharmacologyBiomolecular Engineering