An expeditious synthesis of a biscyclam with an aromatic linker

Nitrogen analogs of crown ethers

Jack E. Richman, Thomas J. Atkins · Journal of the American Chemical Society · 1974 · 636 citations

Natural Sciences, Chemistry, Analytical Chemistry +5

Synthesis and Structure-Activity Relationships of Phenylenebis(methylene)-Linked Bis-Tetraazamacrocycles That Inhibit HIV Replication. Effects of Macrocyclic Ring Size and Substituents on the Aromatic Linker

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Pharmacy, Medicinal Chemistry, Pharmacology +14

Ethyl trifluoroacetate: a powerful reagent for differentiating amino groups

Daqiang Xu, Kapa Prasad, Oljan Repič et al. · Tetrahedron Letters · 1995 · 73 citations

Natural Sciences, Biochemistry, Chemistry +8

Stoichiometric Mono <i>N</i>‐Functionalization of Tetraazamacrocycles via Phosphoryl‐Protected Intermediates

Jean‐Jacques Yaouanc, Henri Handel · Angewandte Chemie International Edition in English · 1991 · 68 citations

Natural Sciences, Chemistry, Organic Chemistry +8

General route for the synthesis of mono N-alkylated derivatives of tetraazamacrocycles

H. BERNARD, Jean‐Jacques Yaouanc, Jean‐Christophe Clément et al. · Tetrahedron Letters · 1991 · 54 citations

Natural Sciences, Chemistry, Medicinal Chemistry +7