Concepedia

Design of novel nicotinic ligands through 3D database searching

Luca Guandalini, Elisabetta Martini, Silvia Dei, Dina Manetti, Serena Scapecchi, Elisabetta Teodori, María Novella Romanelli, Katia Varani, Giovanni Greco, Loredana Spadola,

Bioorganic & Medicinal Chemistry · 2004 · 14 citations · 24 references

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References

24

Crystal structure of an ACh-binding protein reveals the ligand-binding domain of nicotinic receptors

Katjuša Brejc, Willem J. van Dijk, Remco V. Klaassen et al. · Nature · 2001 · 1.8K citations

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A subtype of nicotinic cholinergic receptor in rat brain is composed of alpha 4 and beta 2 subunits and is up-regulated by chronic nicotine treatment.

C M Flores, S W Rogers, L A Pabreza et al. · Molecular Pharmacology · 1992 · 875 citations

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Nicotine and Carbamylcholine Binding to Nicotinic Acetylcholine Receptors as Studied in AChBP Crystal Structures

Patrick H. N. Celie, Sarah E. van Rossum-Fikkert, Willem J. van Dijk et al. · Neuron · 2004 · 775 citations · Full text

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A glia-derived acetylcholine-binding protein that modulates synaptic transmission

August B. Smit, Naweed I. Syed, Dick Schaap et al. · Nature · 2001 · 567 citations

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Cation−π Interactions in Ligand Recognition by Serotonergic (5-HT<sub>3A</sub>) and Nicotinic Acetylcholine Receptors:  The Anomalous Binding Properties of Nicotine

Darren L. Beene, Gabriel S. Brandt, Wenge Zhong et al. · Biochemistry · 2002 · 303 citations

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