Quantitative analysis of racecadotril metabolite in human plasma using a liquid chromatography/tandem mass spectrometry

Pharmacological properties of acetorphan, a parenterally active "enkephalinase" inhibitor.

J Lecomte, Jean Costentin, Adina Vlaiculescu et al. · Journal of Pharmacology and Experimental Therapeutics · 1986 · 144 citations

Medicine, Neuroscience, Pharmacology +13

Racecadotril demonstrates intestinal antisecretory activity in vivo

Marie‐Pierre Primi, Lionel Buéno, P. Bäumer et al. · Alimentary Pharmacology & Therapeutics · 1999 · 72 citations

Medicine, Pharmacology, Pharmacotherapy +14

Enantiomers of thiorphan and acetorphan: correlation between enkephalinase inhibition, protection of endogenous enkephalins and behavioral effects.

Bruno Giros, Claude P. Gros, J.C. Schwartz et al. · Journal of Pharmacology and Experimental Therapeutics · 1987 · 37 citations

Medicine, Medicinal Chemistry, Pharmacology +10

Evaluation of enkephalinase inhibition in the living mouse, using [3H]acetorphan as a probe.

Sophie De La Baume, François Brion, M. Dam Trung Tuong et al. · Journal of Pharmacology and Experimental Therapeutics · 1988 · 17 citations

Medicine, Medicinal Chemistry, Pharmacology +12