Concepedia

Synthesis and structure–activity relationship of 2-(aminoalkyl)-3,3a,8,12b-tetrahydro-2H-dibenzocyclohepta[1,2-b]furan derivatives: a novel series of 5-HT2A/2C receptor antagonists

José M. Cid, José Manuel Alonso Segura, José Ignacio Andrés, Javier Fernández, Pilar Gil, Laura Iturrino, Encarna Matesanz, Theo Meert, Anton Megens, Victor K. Sipido,

Bioorganic & Medicinal Chemistry Letters · 2004 · 19 citations · 16 references

DOIFull text

Open access

Concepts

References

16

[3H]Ketanserin (R 41 468), a selective 3H-ligand for serotonin2 receptor binding sites. Binding properties, brain distribution, and functional role.

J E Leysen, C. J. E. Niemegeers, Jan M. Van Nueten et al. · Molecular Pharmacology · 1982 · 1.1K citations

, , +17

The binding of serotonergic ligands to the porcine choroid plexus: Characterization of a new type of serotonin recognition site

Ángel Pazos, Daniël Hoyer, José Palacios · European Journal of Pharmacology · 1984 · 598 citations

, , +17

Efficacious modification of the mitsunobu reaction for inversions of sterically hindered secondary alcohols

Stephen F. Martin, Jeffrey A. Dodge · Tetrahedron Letters · 1991 · 357 citations

, , +2

Influence of the 5-HT2C receptor antagonist, SB-242084, in tests of anxiety

James R. Martin, Theresa M. Ballard, Guy A. Higgins · Pharmacology Biochemistry and Behavior · 2002 · 140 citations

, , +11

Transferring iodine: more than a simple functional group exchange in organic synthesis

José Barluenga · Pure and Applied Chemistry · 1999 · 116 citations · Full text

, , +2