Automated synthesis of 16α-[18F]fluoroestradiol-3,17β-disulphamate

Sulfamates of various estrogens are prodrugs with increased systemic and reduced hepatic estrogenicity at oral application

W. Elger, Sigfrid Schwarz, Annemarie Hedden et al. · The Journal of Steroid Biochemistry and Molecular Biology · 1995 · 156 citations

Life Sciences, Medicinal Chemistry, Pharmacology +10

The use of 3-methoxymethyl-16β, 17β-epiestriol-O-cyclic sulfone as the precursor in the synthesis of F-18 16α-fluoroestradiol

Jean-Luc Lim, Lei Zheng, Marc S. Berridge et al. · Nuclear Medicine and Biology · 1996 · 78 citations

Life Sciences, Chemistry, Pharmacology +8

Automated production of 16α-[18F]fluoroestradiol for breast cancer imaging

J. Römer, F. Füchtner, Jörg Steinbach et al. · Nuclear Medicine and Biology · 1999 · 49 citations

Medicine, Nuclear Medicine, Oncology +8

Studies on the synthesis of 16α-[18F]fluoroestradiol

Johannes Römer, Jörg Steinbach, H. Kasch · Applied Radiation and Isotopes · 1996 · 35 citations

Medicine, Endocrinology, Pharmacology +6

Steroid sulphatase inhibitors: A new endocrine therapy

M. J. Reed, A Purohit, Nicola M. Howarth et al. · Drugs of the Future · 1984 · 34 citations

Life Sciences, Endocrinology, Pharmacology +14