An efficient and clean CuI-catalyzed chalcogenylation of aromatic azaheterocycles with dichalcogenides

New Arylthioindoles:  Potent Inhibitors of Tubulin Polymerization. 2. Structure−Activity Relationships and Molecular Modeling Studies

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Pharmacy, Medicinal Chemistry, Pharmacology +17

Arylthioindoles, Potent Inhibitors of Tubulin Polymerization

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Medicine, Medicinal Chemistry, Pharmacology +11

5-Chloro-3-(phenylsulfonyl)indole-2-carboxamide: a novel, non-nucleoside inhibitor of HIV-1 reverse transcriptase

Theresa M. Williams, Terrence M. Ciccarone, Suzanne C. MacTough et al. · Journal of Medicinal Chemistry · 1993 · 267 citations · Full text

Medicine, Chemistry, Pharmacology +13

Structural Requirements for Eszopiclone and Zolpidem Binding to the γ-Aminobutyric Acid Type-A (GABA_A) Receptor Are Different

Susan M. Hanson, Elaine V. Morlock, Kenneth A. Satyshur et al. · Journal of Medicinal Chemistry · 2008 · 202 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17

Development of a Novel, Highly Efficient Halide-Catalyzed Sulfenylation of Indoles

Matthew T. Tudge, Minoru Tamiya, Cécile Savarin et al. · Organic Letters · 2006 · 194 citations

Natural Sciences, Chemistry, Medicinal Chemistry +11