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Synthesis and structure–activity relationship of 2-(aminoalkyl)-2,3,3a,8-tetrahydrodibenzo[c,f]isoxazolo[2,3-a]azepine derivatives: a novel series of 5-HT2A/2C receptor antagonists. Part 1

José Ignacio Andrés, Jesús Alcázar, José Manuel Alonso Segura, Javier Fernández, Pilar Gil, Laura Iturrino, Encarna Matesanz, Theo Meert, Anton A. H. P. Megens, Victor K. Sipido

Bioorganic & Medicinal Chemistry Letters · 2002 · 42 citations · 30 references

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30

[3H]Ketanserin (R 41 468), a selective 3H-ligand for serotonin2 receptor binding sites. Binding properties, brain distribution, and functional role.

J E Leysen, C. J. E. Niemegeers, Jan M. Van Nueten et al. · Molecular Pharmacology · 1982 · 1.1K citations

, , +17

The binding of serotonergic ligands to the porcine choroid plexus: Characterization of a new type of serotonin recognition site

Ángel Pazos, Daniël Hoyer, José Palacios · European Journal of Pharmacology · 1984 · 598 citations

, , +17

Serotonin function in anxiety

Dennis S. Charney, Scott W. Woods, Wayne K. Goodman et al. · Psychopharmacology · 1987 · 462 citations

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Serotonergic Responsivity in Obsessive-Compulsive Disorder

Joseph Zohar · Archives of General Psychiatry · 1988 · 295 citations

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Anxiogenic-like effects of mCPP and TFMPP in animal models are opposed by 5-HT1C receptor antagonists

G.A. Kennett, Peter S. Whitton, K. Shah et al. · European Journal of Pharmacology · 1989 · 283 citations

, , +4