Concepedia

(−)-Menthylamine derivatives as potent and selective antagonists of transient receptor potential melastatin type-8 (TRPM8) channels

Giorgio Ortar, Luciano De Petrocellis, Ludovica Morera, Aniello Schiano Moriello, Pierangelo Orlando, Enrico Morera, Marianna Nalli, Vincenzo Di Marzo

Bioorganic & Medicinal Chemistry Letters · 2010 · 35 citations · 12 references

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References

12

Analgesia Mediated by the TRPM8 Cold Receptor in Chronic Neuropathic Pain

Clare J. Proudfoot, Emer M. Garry, David F. Cottrell et al. · Current Biology · 2006 · 413 citations · Full text

, , +13

TRPM8 Mechanism of Cold Allodynia after Chronic Nerve Injury

Hong Xing, Meng Chen, Jennifer Ling et al. · Journal of Neuroscience · 2007 · 222 citations

, , +17

Conservation of Functional and Pharmacological Properties in the Distantly Related Temperature Sensors TRPV1 and TRPM8

Annette Weil, Stephen E. Moore, Nicola J. Waite et al. · Molecular Pharmacology · 2005 · 161 citations

, , +17

Characterisation of TRPM8 as a pharmacophore receptor

Matthias Bödding, Ulrich Wissenbach, Veit Flockerzi · Cell Calcium · 2007 · 128 citations

, , +12

Transient Receptor Potential Channels in Sensory Neurons Are Targets of the Antimycotic Agent Clotrimazole

Víctor Meseguer, Yuji Karashima, Karel Talavera et al. · Journal of Neuroscience · 2008 · 110 citations · Full text

, , +17