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Discovery of novel pyrazolopyrimidinone analogs as potent inhibitors of phosphodiesterase type-5

Sanghapal D. Sawant, G. Lakshma Reddy, Mohd Ishaq Dar, M. Srinivas, Gourav Gupta, Promod Kumar Sahu, Priya Mahajan, Amit Nargotra, Surjeet Singh, S. C. Sharma,

Bioorganic & Medicinal Chemistry · 2015 · 28 citations · 18 references

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18

Glide:  A New Approach for Rapid, Accurate Docking and Scoring. 1. Method and Assessment of Docking Accuracy

Richard A. Friesner, Jay L. Banks, Robert B. Murphy et al. · Journal of Medicinal Chemistry · 2004 · 9.9K citations

, , +17

Glide:  A New Approach for Rapid, Accurate Docking and Scoring. 2. Enrichment Factors in Database Screening

Thomas A. Halgren, Robert B. Murphy, Richard A. Friesner et al. · Journal of Medicinal Chemistry · 2004 · 5.2K citations

, , +17

Sildenafil: an orally active type 5 cyclic GMP-specific phosphodiesterase inhibitor for the treatment of penile erectile dysfunction.

Mitra Boolell, Allen Mj, Ballard Sa et al. · PubMed · 1996 · 1.1K citations

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Sildenafil (VIAGRATM), a potent and selective inhibitor of type 5 cGMP phosphodiesterase with utility for the treatment of male erectile dysfunction

N.K. Terrett, Andrew Bell, David Brown et al. · Bioorganic & Medicinal Chemistry Letters · 1996 · 606 citations

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Pharmacokinetics and metabolism of sildenafil in mouse, rat, rabbit, dog and man

Don K. Walker · Xenobiotica · 1999 · 401 citations

, , +16