Concepedia

Discovery of selective dopamine D4 receptor antagonists: 1-Aryloxy-3-(4-aryloxypiperidinyl)-2-propanols

Jon L. Wright, Tracy F. Gregory, Thomas G. Heffner, Robert G. MacKenzie, Thomas A. Pugsley, Seth Vander Meulen, Lawrence D. Wise

Bioorganic & Medicinal Chemistry Letters · 1997 · 35 citations · 5 references

DOI

Concepts

References

5

Cloning of the gene for a human dopamine D4 receptor with high affinity for the antipsychotic clozapine

Hubert H.M. Van Tol, James R. Bunzow, Hong‐Chang Guan et al. · Nature · 1991 · 2K citations · Full text

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Neurochemical and functional characterization of the preferentially selective dopamine D3 agonist PD 128907.

Thomas A. Pugsley, M. Duff Davis, Hyacinth C. Akunne et al. · Journal of Pharmacology and Experimental Therapeutics · 1995 · 201 citations

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Full-length cDNA cloning and distribution of human dopamine D4 receptor

Mitsuyuki Matsumoto, Kazuyuki Hidaka, Shoko Tada et al. · Molecular Brain Research · 1995 · 140 citations

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D2 dopamine receptor stimulation of mitogenesis in transfected Chinese hamster ovary cells: relationship to dopamine stimulation of tyrosine phosphorylations.

Mary E. Lajiness, Chris L. Chio, Rita M. Huff · Journal of Pharmacology and Experimental Therapeutics · 1993 · 62 citations

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The Discovery and Structure-Activity Relationships of 1,2,3,6-Tetrahydro-4-phenyl-1-[(arylcyclohexenyl)alkyl]pyridines. Dopamine Autoreceptor Agonists and Potential Antipsychotic Agents

Jon L. Wright, Bradley W. Caprathe, Dennis M. Downing et al. · Journal of Medicinal Chemistry · 1994 · 26 citations · Full text

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