Concepedia

Comparative Alpha-1 Adrenoceptor Subtype Selectivity and Functional Uroselectivity of Alpha-1 Adrenoceptor Antagonists

Denis Martin, Philippe Lluel, Etienne Guillot, A. Coste, D Jammes, I. Angel

Journal of Pharmacology and Experimental Therapeutics · 1997 · 88 citations · 26 references

DOI

Concepts

References

26

The alpha 1-adrenergic receptor that mediates smooth muscle contraction in human prostate has the pharmacological properties of the cloned human alpha 1c subtype.

Carlos Forray, Jonathan Bard, J. M. WETZEL et al. · Molecular Pharmacology · 1994 · 349 citations

, , +13

Identification, Quantification, and Localization of mRNA for Three Distinct Alpha<sub>1</sub>Adrenergic Receptor Subtypes in Human Prostate

David T. Price, Debra A. Schwinn, Jon W. Lomasney et al. · The Journal of Urology · 1993 · 322 citations

, , +7

RS-17053 (N-[2-(2-cyclopropylmethoxyphenoxy)ethyl]-5-chloro-alpha, alpha-dimethyl-1H-indole-3-ethanamine hydrochloride), a selective alpha 1A-adrenoceptor antagonist, displays low affinity for functional alpha 1-adrenoceptors in human prostate: implications for adrenoceptor classification.

Anthony Ford, Nicolas F. Arredondo, David R. Blue et al. · Molecular Pharmacology · 1996 · 193 citations

, , +13

Noradrenaline contractions of human prostate mediated by α<sub>1c</sub>‐(α<sub>1c</sub>‐) adrenoceptor subtype

Ian Marshall, Richard P. Burt, C.R. Chappie · British Journal of Pharmacology · 1995 · 155 citations · Full text

, , +9

In vitro characterization of the α-adrenoceptors in human prostate

J. Paul Hieble, Marco Caine, Ety Zalaznik · European Journal of Pharmacology · 1985 · 145 citations

, , +7