Heterocycles. VI. Syntheses of 4H-s-Triazolo [4, 3-a] [1, 4] benzodiazepines, Novel Tricyclic Psychosedatives

Kanji Meguro, H. TAWADA, Hiroshi Miyano, Yoshiaki Sato, Y. KUWADA

Chemical and Pharmaceutical Bulletin · 1973 · 26 citations · 0 references

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Abstract

A variety of 4H-s-triazolo [4, 3-a] [1, 4] benzodiazepines (VII) which are highly active in central nervous system depression was synthesized with the aim of investigating structure-activity relationships.