Optimization of on-resin palladium-catalyzed Sonogashira cross-coupling reaction for peptides and its use in a structure–activity relationship study of a class B GPCR ligand

Copper-Free Sonogashira Cross-Coupling for Functionalization of Alkyne-Encoded Proteins in Aqueous Medium and in Bacterial Cells

Nan Li, Reyna K. V. Lim, Selvakumar Edwardraja et al. · Journal of the American Chemical Society · 2011 · 262 citations · Full text

Natural Sciences, Biochemistry, Chemistry +13

Proline Editing: A General and Practical Approach to the Synthesis of Functionally and Structurally Diverse Peptides. Analysis of Steric versus Stereoelectronic Effects of 4-Substituted Prolines on Conformation within Peptides

Anil K. Pandey, Devan Naduthambi, Krista Thomas et al. · Journal of the American Chemical Society · 2013 · 177 citations

Life Sciences, Biochemistry, Medicinal Chemistry +15

Phthalocyanine–Peptide Conjugates: Receptor-Targeting Bifunctional Agents for Imaging and Photodynamic Therapy

Elena Ranyuk, Nicole Cauchon, Klaus Klarskov et al. · Journal of Medicinal Chemistry · 2013 · 116 citations

Medicine, Medicinal Chemistry, Pharmacology +17

Bioconjugation of Peptides by Palladium-Catalyzed C−C Cross-Coupling in Water

Harald Dibowski, Franz P. Schmidtchen · Angewandte Chemie International Edition · 1998 · 102 citations

Natural Sciences, Biochemistry, Chemistry +15

Class-B GPCR activation: is ligand helix-capping the key?

Jean‐Michel Neumann, Alain Couvineau, Samuel Murail et al. · Trends in Biochemical Sciences · 2008 · 98 citations

Life Sciences, Biochemistry, Molecular Biology +12