Synthesis and antiplasmodial activity of new 4-aryl-2-trichloromethylquinazolines

Pierre Verhaeghe, Nadine Azas, M. Gasquet, +6

Bioorganic & Medicinal Chemistry Letters

HeterocyclicAntiplasmodial ActivityOrganic ChemistryChemistryHeterocycle Chemistry +2

New aromatase inhibitors. Synthesis and biological activity of aryl-substituted pyrrolizine and indolizine derivatives

Pascal Sonnet, Patrick Dallemagne, Jean Guillon, +9

Bioorganic & Medicinal Chemistry

BiochemistryMedicineAryl-substituted PyrrolizineAromataseNew Aromatase Inhibitors +5

Synthesis and Structure–Affinity Relationships of Selective High-Affinity 5-HT₄Receptor Antagonists: Application to the Design of New Potential Single Photon Emission Computed Tomography Tracers

Emmanuelle Dubost⧫, Noé Dumas, Christine Fossey, +11

Journal of Medicinal Chemistry

Reactivity of 3-Iodoimidazo[1,2-<i>a</i>]pyridines Using a Suzuki-Type Cross-Coupling Reaction

Cécile Enguehard‐Gueiffier, Jean‐Louis Renou, Valérie Collot, +3

The Journal of Organic Chemistry

Strong BasesChemical EngineeringCross-coupling ReactionSuzuki Cross-coupling ReactionEngineering +5

Synthesis of novel halopyridinylboronic acids and esters. Part 4: Halopyridin-2-yl-boronic acids and esters are stable, crystalline partners for classical Suzuki cross-coupling

Alexandre Bouillon, Jean‐Charles Lancelot, Jana Sopková‐de Oliveira Santos, +3

Tetrahedron

Cross-coupling ReactionEngineeringNovel Halopyridinylboronic AcidsOrganic ChemistryClassical Suzuki Cross-coupling +5

Synthesis of novel halopyridinylboronic acids and esters. Part 1: 6-Halopyridin-3-yl-boronic acids and esters

Alexandre Bouillon, Jean‐Charles Lancelot, Valérie Collot, +2

Tetrahedron

EngineeringNovel Halopyridinylboronic AcidsOrganic ChemistryChemistry6-Halopyridin-3-yl-boronic Acids +4

Synthesis of new pyrrolo[1,2-a]quinoxalines: potential non-peptide glucagon receptor antagonists

Jean Guillon, Patrick Dallemagne, Bruno Pfeiffer, +4

European Journal of Medicinal Chemistry

Molecular PharmacologyMedicinal ChemistryMedicineHeterocycle ChemistryPharmacology +2

Toward Safer Thrombolytic Agents in Stroke: Molecular Requirements for NMDA Receptor-Mediated Neurotoxicity

José P. López‐Atalaya, Benoit D. Roussel, Denis Levrat, +14

Journal of Cerebral Blood Flow & Metabolism

Suzuki-type cross-coupling reaction of 3-iodoindazoles with aryl boronic acids: A general and flexible route to 3-arylindazoles

Valérie Collot, Patrick Dallemagne, Philippe R. Bovy, +1

Tetrahedron

Cross-coupling ReactionEngineeringAryl Boronic AcidsSuzuki-type Cross-coupling ReactionOrganic Chemistry +4

Effect of A-Ring Modifications on the DNA-Binding Behavior and Cytotoxicity of Pyrrolo[2,1-<i>c</i>][1,4]benzodiazepines

David E. Thurston, D. Subhas Bose, Philip W. Howard, +8

Journal of Medicinal Chemistry

Combinatorial ChemistryBioorganic ChemistryPyrimidine RingsPharmacotherapyHeterocycle Chemistry +18