Jean-Claude Brelière

In vitro and in vivo biological activities of SR140333, a novel potent non-peptide tachykinin NK1 receptor antagonist

Xavier Emonds‐Alt, Jean-Daniel Doutremepuich, Michel Héaulme et al. · European Journal of Pharmacology · 1993 · 374 citations

Pharmacy, Medicinal Chemistry, Pharmacology +5

Biochemical and pharmacological characterisatioN OF SR141716A, the first potent and selective brain cannabinoid receptor antagonist

Murielle Rinaldi‐Carmona, Francis Barth, Michel Héaulme et al. · Life Sciences · 1995 · 300 citations

Medicine, Neuroscience, Pharmacology +10

Characterization and distribution of binding sites for [3H]-SR 141716A, a selective brain (CB1) cannabinoid receptor antagonist, in rodent brain

Murielle Rinaldi‐Carmona, Françoise Pialot, Christian Congy et al. · Life Sciences · 1996 · 131 citations

Medicine, Neuroscience, Pharmacology +12

Effects on the Isolated Human Bronchus of SR 48968, a Potent and Selective Nonpeptide Antagonist of the Neurokinin A (NK2) Receptors

Charles Advenier, Emmanuel Naline, Lucien Toty et al. · American Review of Respiratory Disease · 1992 · 109 citations

Medicine, Pharmacology, Cancer Pharmacology +8

A new series of imidazolones: highly specific and potent nonpeptide AT1 angiotensin II receptor antagonists

C. BERNHART, Pierre Perreaut, Yvette Muneaux et al. · Journal of Medicinal Chemistry · 1993 · 108 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16