New Pyrrole Inhibitors of Monoamine Oxidase:  Synthesis, Biological Evaluation, and Structural Determinants of MAO-A and MAO-B Selectivity

Giuseppe La Regina, Romano Silvestri, Marino Artico, +5

Journal of Medicinal Chemistry

Combinatorial ChemistryOrganic ChemistryPharmacotherapyChemistryChemical Biology +18

Quercetin as the Active Principle of<i>Hypericum</i><i>h</i><i>ircinum</i>Exerts a Selective Inhibitory Activity against MAO-A:  Extraction, Biological Analysis, and Computational Study

Franco Chimenti, Filippo Cottiglia, Leonardo Bonsignore, +14

Journal of Natural Products

Synthesis, Molecular Modeling Studies, and Selective Inhibitory Activity against Monoamine Oxidase of 1-Thiocarbamoyl-3,5-diaryl-4,5-dihydro-(1<i>H</i>)- pyrazole Derivatives

Franco Chimenti, Elias Maccioni, Daniela Secci, +11

Journal of Medicinal Chemistry

Synthesis and Selective Inhibitory Activity of 1-Acetyl-3,5-diphenyl-4,5-dihydro-(1<i>H</i>)-pyrazole Derivatives against Monoamine Oxidase

Franco Chimenti, Adriana Bolasco, Fedele Manna, +8

Journal of Medicinal Chemistry

Inhibition of monoamine oxidases by coumarin-3-acyl derivatives: biological activity and computational study

Franco Chimenti, Daniela Secci, Adriana Bolasco, +6

Bioorganic & Medicinal Chemistry Letters

Biological ActivityCoumarin-3-acyl DerivativesPharmacological StudyBiochemistryMedicine +7

Inhibition of amine oxidases activity by 1-acetyl-3,5-diphenyl-4,5-dihydro-(1H)-pyrazole derivatives

Fedele Manna, Franco Chimenti, Adriana Bolasco, +7

Bioorganic & Medicinal Chemistry Letters

Medicinal ChemistryBiochemistryNatural SciencesHeterocycle ChemistryPharmacology +3

Selective Inhibitory Activity against MAO and Molecular Modeling Studies of 2-Thiazolylhydrazone Derivatives

Franco Chimenti, Elias Maccioni, Daniela Secci, +9

Journal of Medicinal Chemistry

Bioorganic ChemistryMao-b IsoformsOrganic ChemistryPharmacotherapyMedicinal Chemistry +15

Purification of bovine plasma amine oxidase

Paola Turini, Stefania Sabatini, Olivia Befani, +3

Analytical Biochemistry

Purification MethodBiotechnologyBiochemistryProtein Purification

Monoamine Oxidase Isoform-Dependent Tautomeric Influence in the Recognition of 3,5-Diaryl Pyrazole Inhibitors

Franco Chimenti, Rossella Fioravanti, Adriana Bolasco, +7

Journal of Medicinal Chemistry

Medicinal ChemistryMonoamine Oxidase BBioorganic ChemistryTautomeric EquilibriaBiochemistry +13

Enzymatic oxidation products of spermine induce greater cytotoxic effects on human multidrug‐resistant colon carcinoma cells (LoVo) than on their wild‐type counterparts

Annarica Calcabrini, Giuseppe Arancia, Manuela Marra, +4

International Journal of Cancer