David Tien

A simple procedure for the solid phase synthesis of diketopiperazine and diketomorpholine derivatives

Anna Katrin Szardenings, Timothy S. Burkoth, Henry H. Lu et al. · Tetrahedron · 1997 · 129 citations

Combinatorial Chemistry, Derivative (Chemistry), Diketomorpholine Derivatives +7

Identification of Highly Selective Inhibitors of Collagenase-1 from Combinatorial Libraries of Diketopiperazines

Anna Katrin Szardenings, Valery V. Antonenko, David A. Campbell et al. · Journal of Medicinal Chemistry · 1999 · 66 citations · Full text

Highly Selective Inhibitors, Medicinal Chemistry, Drug Target +15

Rational Design and Combinatorial Evaluation of Enzyme Inhibitor Scaffolds:  Identification of Novel Inhibitors of Matrix Metalloproteinases

Anna Katrin Szardenings, David C.H. Harris, Stuart Lam et al. · Journal of Medicinal Chemistry · 1998 · 57 citations · Full text

Combinatorial Libraries, Chemical Biology, Pharmaceutical Chemistry +18

Malonyl α-mercaptoketones and α-mercaptoalcohols, a new class of matrix metalloproteinase inhibitors

David A. Campbell, Xiao-Yi Xiao, David C.H. Harris et al. · Bioorganic & Medicinal Chemistry Letters · 1998 · 24 citations · Full text

Biochemistry, Malonyl α-Mercaptoketones, Medicine +9