Tetsuya Sekiguchi

Discovery of Gemilukast (ONO-6950), a Dual CysLT₁and CysLT₂Antagonist As a Therapeutic Agent for Asthma

Satoshi Itadani, Kentaro Yashiro, Yoshiyuki Aratani et al. · Journal of Medicinal Chemistry · 2015 · 24 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Discovery of novel S1P2 antagonists, part 3: Improving the oral bioavailability of a series of 1,3-bis(aryloxy)benzene derivatives

Kensuke Kusumi, Koji Shinozaki, Yoshiyuki Yamaura et al. · Bioorganic & Medicinal Chemistry Letters · 2016 · 21 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +14

Discovery of novel S1P2 antagonists. Part 1: Discovery of 1,3-bis(aryloxy)benzene derivatives

Kensuke Kusumi, Koji Shinozaki, Toshiya Kanaji et al. · Bioorganic & Medicinal Chemistry Letters · 2015 · 18 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Discovery of novel S1P2 antagonists. Part 2: Improving the profile of a series of 1,3-bis(aryloxy)benzene derivatives

Kensuke Kusumi, Koji Shinozaki, Yoshiyuki Yamaura et al. · Bioorganic & Medicinal Chemistry Letters · 2015 · 17 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +12

Discovery of Highly Potent Dual CysLT₁ and CysLT₂ Antagonist

Satoshi Itadani, Shinya Takahashi, Masaki Ima et al. · ACS Medicinal Chemistry Letters · 2014 · 15 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +9