Musong Kim

2,4,6-Triaminopyrimidine as a Novel Hinge Binder in a Series of PI3Kδ Selective Inhibitors

Leena Patel, Jayaraman Chandrasekhar, Jerry Evarts et al. · Journal of Medicinal Chemistry · 2016 · 47 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Discovery of Orally Efficacious Phosphoinositide 3-Kinase δ Inhibitors with Improved Metabolic Stability

Leena Patel, Jayaraman Chandrasekhar, Jerry Evarts et al. · Journal of Medicinal Chemistry · 2016 · 46 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +15

The In Vitro Pharmacology of GS-5759, A Novel Bifunctional Phosphodiesterase 4 Inhibitor and Long Acting β2-Adrenoceptor Agonist

Stacey Tannheimer, Eric A. Sorensen, Zhi-Hua Cui et al. · Journal of Pharmacology and Experimental Therapeutics · 2014 · 29 citations

Medicine, Medicinal Chemistry, Pharmacology +16

The in vivo efficacy and side effect pharmacology of <scp>GS</scp>‐5759, a novel bifunctional phosphodiesterase 4 inhibitor and long‐acting <i>β</i>₂‐adrenoceptor agonist in preclinical animal species

M Salmon, Stacey Tannheimer, Terry T. Gentzler et al. · Pharmacology Research & Perspectives · 2014 · 19 citations · Full text

Medicine, Pharmacology, Pharmacotherapy +14

GS-5759, a Bifunctional β2-Adrenoceptor Agonist and Phosphodiesterase 4 Inhibitor for Chronic Obstructive Pulmonary Disease with a Unique Mode of Action: Effects on Gene Expression in Human Airway Epithelial Cells

Taruna Joshi, Omar Hamed, Stacey Tannheimer et al. · Journal of Pharmacology and Experimental Therapeutics · 2016 · 19 citations

Medicine, Medicinal Chemistry, Pharmacology +17