Marcin Leś

Lithocholic Acid Hydroxyamide Destabilizes Cyclin D1 and Induces G 0 /G 1 Arrest by Inhibiting Deubiquitinase USP2a

Katarzyna Magiera‐Mularz, Marcin D. Tomala, Katarzyna Kubica et al. · Cell chemical biology · 2017 · 57 citations · Full text

Medicine, Cancer Biology, Oncology +17

Synthesis of amide and sulfonamide substituted N-aryl 6-aminoquinoxalines as PFKFB3 inhibitors with improved physicochemical properties

Nicolas Boutard, Arkadiusz Białas, Aleksandra Sabiniarz et al. · Bioorganic & Medicinal Chemistry Letters · 2018 · 24 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +10

Discovery and Structure–Activity Relationships of <i>N</i>‐Aryl 6‐Aminoquinoxalines as Potent PFKFB3 Kinase Inhibitors

Nicolas Boutard, Arkadiusz Białas, Aleksandra Sabiniarz et al. · ChemMedChem · 2018 · 21 citations · Full text

Life Sciences, Medicinal Chemistry, Pharmacology +17

Discovery of 5-{2-[5-Chloro-2-(5-ethoxyquinoline-8-sulfonamido)phenyl]ethynyl}-4-methoxypyridine-2-carboxylic Acid, a Highly Selective in Vivo Useable Chemical Probe to Dissect MCT4 Biology

Timo Heinrich, Ada Sala-Hojman, Roberta Ferretti et al. · Journal of Medicinal Chemistry · 2021 · 21 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +16