Po‐Chu Kuo

Optimization of Ligand and Lipophilic Efficiency To Identify an in Vivo Active Furano-Pyrimidine Aurora Kinase Inhibitor

Hui‐Yi Shiao, Mohane Selvaraj Coumar, Chang Chun-Wei et al. · Journal of Medicinal Chemistry · 2013 · 41 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17

Discovery of 1-(2,4-Dichlorophenyl)-<i>N</i>-(piperidin-1-yl)-4-((pyrrolidine-1-sulfonamido)methyl)-5-(5-((4-(trifluoromethyl)phenyl)ethynyl)thiophene-2-yl)-1<i>H</i>-pyrazole-3-carboxamide as a Novel Peripherally Restricted Cannabinoid-1 Receptor Antagonist with Significant Weight-Loss Efficacy in Diet-Induced Obese Mice

Chun‐Ping Chang, Chien-Huang Wu, Jen‐Shin Song et al. · Journal of Medicinal Chemistry · 2013 · 36 citations

Pharmacy, Medicinal Chemistry, Pharmacology +13

Design, Synthesis, and Evaluation of Thiazolidine-2,4-dione Derivatives as a Novel Class of Glutaminase Inhibitors

Teng‐Kuang Yeh, Ching‐Chuan Kuo, Yue‐Zhi Lee et al. · Journal of Medicinal Chemistry · 2017 · 32 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +13

Discovery of 1‐(2,4‐Dichlorophenyl)‐4‐ethyl‐5‐(5‐(2‐(4‐(trifluoromethyl)phenyl)ethynyl)thiophen‐2‐yl)‐<i>N</i>‐(piperidin‐1‐yl)‐1<i>H</i>‐pyrazole‐3‐carboxamide as a Potential Peripheral Cannabinoid‐1 Receptor Inverse Agonist

Ming‐Shiu Hung, Chun‐Ping Chang, T. LI et al. · ChemMedChem · 2010 · 25 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +11

Development of Stem-Cell-Mobilizing Agents Targeting CXCR4 Receptor for Peripheral Blood Stem Cell Transplantation and Beyond

Chien-Huang Wu, Jen‐Shin Song, Hsuan-Hao Kuan et al. · Journal of Medicinal Chemistry · 2018 · 19 citations · Full text

Pharmacy, Medicinal Chemistry, Pharmacology +17