Sam Lawn

Computer-aided drug discovery of Myc-Max inhibitors as potential therapeutics for prostate cancer

Lavinia A. Carabet, Nada Lallous, Eric Leblanc et al. · European Journal of Medicinal Chemistry · 2018 · 58 citations · Full text

Medicine, Medicinal Chemistry, Oncology +13

Discovery and characterization of small molecules targeting the DNA-binding ETS domain of ERG in prostate cancer

Miriam Butler, Mani Roshan‐Moniri, Michael Hsing et al. · Oncotarget · 2017 · 45 citations · Full text

Medicine, Molecular Biology, Oncology +12

Targeting Binding Function-3 of the Androgen Receptor Blocks Its Co-Chaperone Interactions, Nuclear Translocation, and Activation

Nada Lallous, Eric Leblanc, Ravi S. N. Munuganti et al. · Molecular Cancer Therapeutics · 2016 · 29 citations · Full text

Medicine, Oncology, Pharmacology +17

In vitro modeling of glioblastoma initiation using PDGF-AA and p53-null neural progenitors

Alexandra Böhm, Jessica DePetro, Carmen Binding et al. · Neuro-Oncology · 2020 · 18 citations · Full text

Life Sciences, Cell Biology, Oncology +16

Development of 2-(5,6,7-Trifluoro-1<i>H</i>-Indol-3-yl)-quinoline-5-carboxamide as a Potent, Selective, and Orally Available Inhibitor of Human Androgen Receptor Targeting Its Binding Function-3 for the Treatment of Castration-Resistant Prostate Cancer

Eric Leblanc, Fuqiang Ban, Ayşe Derya Cavga et al. · Journal of Medicinal Chemistry · 2021 · 15 citations · Full text

Medicine, Medicinal Chemistry, Pharmacology +17